Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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TLK1

RBC: TLK1 · Substrate: Histone H3 ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Bosutinib42.00.55
Defactinib38.50.45
Lapatinib25.00.62
Midostaurin22.80.50
Pacritinib22.00.45
Ponatinib19.80.53
Gilteritinib19.60.51
Ceritinib17.80.62
Mobocertinib16.70.76
Neratinib16.20.60
Pirtobrutinib15.30.66
Tenalisib15.00.70
Lazertinib14.90.67
Capmatinib14.70.58
Crizotinib13.90.58

Known variants

No variants catalogued.
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