CDK2/CCNE2
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Defactinib | 89.9 | 0.45 |
| Abemaciclib | 62.8 | 0.56 |
| Pralsetinib | 53.6 | 0.64 |
| Vemurafenib | 34.2 | 0.60 |
| Pacritinib | 30.4 | 0.45 |
| Repotrectinib | 23.0 | 0.61 |
| Midostaurin | 19.0 | 0.50 |
| Neratinib | 18.4 | 0.60 |
| Gilteritinib | 16.7 | 0.51 |
| Pirtobrutinib | 14.7 | 0.66 |
| Palbociclib | 14.1 | 0.67 |
| Entrectinib | 13.2 | 0.67 |
| Brigatinib | 12.7 | 0.51 |
| Baricitinib | 11.7 | 0.62 |
| Lorlatinib | 11.2 | 0.69 |
Known variants
No variants catalogued.