DYRK4
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Avapritinib | 52.6 | 0.64 |
| Abemaciclib | 21.7 | 0.56 |
| Defactinib | 21.0 | 0.45 |
| Gedatolisib | 13.4 | 0.61 |
| Pirtobrutinib | 10.4 | 0.66 |
| Pacritinib | 9.6 | 0.45 |
| Alectinib | 9.3 | 0.65 |
| Mobocertinib | 8.5 | 0.76 |
| Capivasertib | 8.0 | 0.64 |
| Infigratinib | 7.6 | 0.71 |
| Fostamatinib | 7.6 | 0.61 |
| Tenalisib | 7.5 | 0.70 |
| Ceritinib | 7.4 | 0.62 |
| Neratinib | 7.2 | 0.60 |
| Lapatinib | 6.9 | 0.62 |
Known variants
No variants catalogued.