GRK4
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Alectinib | 71.1 | 0.65 |
| Ceritinib | 42.7 | 0.62 |
| Midostaurin | 19.5 | 0.50 |
| Brigatinib | 18.1 | 0.51 |
| Lorlatinib | 18.0 | 0.69 |
| Darovasertib | 17.8 | 0.72 |
| Entrectinib | 14.4 | 0.67 |
| Capivasertib | 14.4 | 0.64 |
| Quizartinib | 13.9 | 0.74 |
| Canertinib | 13.0 | 0.67 |
| Sunitinib | 11.6 | 0.52 |
| Repotrectinib | 11.0 | 0.61 |
| Nintedanib | 10.6 | 0.61 |
| Alpelisib | 10.0 | 0.72 |
| Crizotinib | 9.8 | 0.58 |
Known variants
No variants catalogued.