Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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MAP3K3

RBC: MEKK3 · Substrate: MBP ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Ponatinib94.10.53
Crizotinib90.30.58
Bosutinib84.10.55
Ripretinib81.50.67
Midostaurin80.20.50
Neratinib78.10.60
Nintedanib76.40.61
Repotrectinib63.30.61
Infigratinib62.50.71
Sunitinib61.20.52
Dasatinib59.40.70
Ruxolitinib57.00.59
Baricitinib55.90.62
Apatinib53.20.70
Pemigatinib52.90.72

Known variants

No variants catalogued.
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