Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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TNK2

RBC: ACK1 · Substrate: Lyntide 2+Mn ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Bosutinib100.00.55
Lorlatinib99.30.69
Repotrectinib99.00.61
Brigatinib98.00.51
Dasatinib97.80.70
Mobocertinib97.40.76
Entrectinib97.30.67
Ceritinib97.20.62
Midostaurin96.90.50
Neratinib95.20.60
Ponatinib94.90.53
Pacritinib94.50.45
Fedratinib93.40.58
Osimertinib92.60.73
Alectinib89.20.65

Known variants

No variants catalogued.
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