Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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PDGFRB

RBC: PDGFRb · Substrate: pEY + Mn ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Ponatinib100.00.53
Nintedanib96.00.61
Tivozanib95.80.67
Regorafenib95.40.72
Axitinib92.90.69
Dasatinib92.50.70
Avapritinib90.40.64
Midostaurin89.90.50
Ripretinib89.10.67
Quizartinib89.00.74
Nilotinib86.70.77
Sunitinib84.80.52
Pralsetinib81.30.64
Apatinib80.90.70
Sorafenib80.80.78

Known variants

No variants catalogued.
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