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Paxalisib

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Primary targets: PI3K, MTOR_FRAP1 · FDA status: FDA Phase III Trials to begin

Selectivity scorecard

KISS
99.75
Gini
0.609
CATDS
0.039

Computed from wild-type kinome inhibition at 1 μM. Gini reproduces the published values within tolerance; KISS and CATDS are computed but pending reconciliation with the paper's reference code.

Polypharmacology radar

Top 20 strongest-inhibited wild-type kinases for Paxalisib. Strongest target: CHK1 at 95.2% inhibition.

Accessible data table
RankTargetInhibition %Residual activity %
1CHK195.2%4.8%
2MTOR_FRAP181.2%18.8%
3RAF154.2%45.8%
4MLK2_MAP3K1046.7%53.3%
5YES_YES142.8%57.2%
6MLK3_MAP3K1138.6%61.4%
7CAMK2D35.8%64.2%
8RSK334.1%65.9%
9LCK29.5%70.5%
10BTK27.1%72.9%
11CDK3_CYCLIN_C26.6%73.4%
12HCK26.0%74.0%
13CAMK2A24.1%75.9%
14PAK422.5%77.5%
15SYK22.3%77.7%
16FLT320.6%79.4%
17BLK20.2%79.8%
18FYN20.2%79.8%
19TXK19.4%80.6%
20FGR19.1%80.9%

Selectivity landscape

Where Paxalisib sits in the 92-drug selectivity landscape (KISS vs Gini). The highlighted point is Paxalisib.

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